Bioorganic and Medicinal Chemistry Letters

Paper

01 Jan 1993

Synthesis of 4(5)-imidazolyl allylamines and propargylamines as inhibitors of diamine oxidase

View publication

Abstract

A series of four side-chain unsaturated histamine analogs were synthesized and evaluated as inhibitors of Diamine Oxidase, (DAO). All four target compounds were potent competitive inhibitors of DAO with Ki values ranging from 0.17 to 7.1 μM. © 1993.

Paper

Transcriptional evidence for the "Reverse Warburg Effect" in human breast cancer tumor stroma and metastasis: Similarities with oxidative stress, inflammation, Alzheimer's disease, and "Neuron-Glia Metabolic Coupling"

Stephanos Pavlides, Aristotelis Tsirigos, et al.

Aging

Paper

Glass microneedles for force measurements: A finite-element analysis model

Peter N. Ayittey, John S. Walker, et al.

Pflugers Archiv European Journal of Physiology

Paper

Determining subunit-subunit interaction from statistics of cryo-EM images: observation of nearest-neighbor coupling in a circadian clock protein complex

Xu Han, Dongliang Zhang, et al.

Nature Communications

Paper

The binding mode of progesterone to its receptor deduced from molecular dynamics simulations

Tiziana Mordasini, Alessandro Curioni, et al.

ChemBioChem

View all publications